Koeke Rongoa Maamaa Teitei 877399-52-5 Crizotinib mo te Tiaki Mate pukupuku
Huaingoa | Crizotinib |
Nga kupu taurite | PF-02341066;3-[(1R)-1-(2,6-Dichloro-3-fluorophenyl)ethoxy]-5-[1-(4-piperidinyl)-1H-pyrazol-4-yl]pyridin-2-amine;PF 2341066 |
CAS No. | 877399-52-5 |
Te ahua | Ma ki te paura tioata ma-kore |
Tātai rāpoi | C21H22Cl2FN5O |
Taumaha rāpoi | 450.34 |
Whakamahinga | Tohu Rongoa, kaupapa Rangahau ranei |
Te takai | Ka rite ki to tono |
Rokiroki | Whakaorangia i roto i nga ipu kiki, kare-marama i te waahi makariri |
CrizotinibCas: 877399-52-5 | ||
Nga taonga | Whakatakotoranga | Hua |
Te ahua | Ma ki te paura tioata ma-kore | Te paura tioata ma |
Tautuhinga | H-NMR, MS | Ka tutuki |
Wairewa toenga | isopropanol≤0.5% EtOAc≤0.5% THF≤0.072% n-Heptane≤0.5% Toluene≤0.5% | 0.3% ND ND ND ND ND |
Nga Korewa Taamaha | ≤10ppm | Ka tutuki |
Te ihirangi wai | £0.5% | 0.3% |
Te toenga i runga i te mura | £0.5% | 0.05% |
Enantiomer | £0.1% | <LOQ |
He poke e pa ana na HPLC | Kotahi poke≤0.1% Te poke katoa ≤1.0% | 0.05% 0.12% |
Pure (HPLC) | ³99.0% | 99.88% |
Nga korero a te Kamupene
√ Ko nga wheako katoa o te paparanga whakahaere i roto i te wheketere me nga kaitoi mohio nga akonga; √ Ko te kounga tonu to maatau whakaaro nui, te punaha QC tino tika; √ 11 tau te mohio ki te kawe i te roopu hoko; √ taiwhanga R&D motuhake; √ E rua nga awheawhe GMP roa kua hainatia; √ He nui nga rawa o nga wheketere mangere mo te kaupapa kua whakaritea; √ He roopu mahi Kairangi me te huarahi rite.Tuhia to korero ki konei ka tukuna mai ki a matou