Koeke Rongoa Maamaa Teitei 1421373-66-1 Mesylate-AZD9291 mo te maimoatanga mate pukupuku
Huaingoa | AZD-9291 mesylate |
Nga kupu taurite | N-[2-[[2-(Dimethylamino)ethyl]methylamino]-4-methoxy-5-[[4-(1-methyl-1H-indol-3-yl)-2-pyrimidinyl]amino]phenyl]- 2-propenamide methanesulfonate (1:1) |
CAS No. | 1421373-66-1 |
Te ahua | Ma ki te kowhai marama te paura totoka |
Tātai rāpoi | C28H33N7O2.CH4O3S |
Taumaha rāpoi | 595.71 |
Whakamahinga | Tohu Rongoa, kaupapa Rangahau ranei |
Te takai | Ka rite ki to tono |
Rokiroki | Whakaorangia i roto i nga ipu kiki, kare-marama i te waahi makariri |
AZD-9291 mesylateCAS:1421373-66-1 | ||
Items | Stohu | Rhua |
Te ahua | Ma ki te kowhai marama te paura totoka | Te paura totoka kowhai marama |
Itohu tohu | Na IR | Ka tutuki |
Na HPLC | Ka tutuki | |
Wairewa | Wairewa i roto i te Dimethylsulfoxide, paku wairewa i roto i te Ethanol me te Acetonitrile, me te wairewa wai e whakawhirinaki ana ki te pH. | Ka tutuki |
Ihirangi wai(KF) | ≤ 1.00% | 0.42% |
Te toenga i runga i te mura | ≤ 0.10% | 0.05% |
HtaumahaMetal | ≤ 20ppm | Ka tutuki |
Mesylate | 15.20%~18.20% | 15.90% |
Wairewa toenga | Acetonitrile: ≤410ppm | ND |
Acetone: ≤5000ppm | ND | |
Tetrahydrofuran: ≤720ppm | ND | |
RkoakoaSmatū | Te nuinga o te poke kotahi: ≤0.20% | 0.17% |
Tapeke poke: ≤1.00% | 0.25% | |
Rahi Matūriki | D90: ≤100μm | 57.97% |
Akorero (HPLC i runga i te whakamaroke) | 98.00%~102.00% | 99.80% |
Paerewa Tohutoro | Paerewa o-whare |
Nga korero a te Kamupene
√ Ko nga wheako katoa o te paparanga whakahaere i roto i te wheketere me nga kaitoi mohio nga akonga; √ Ko te kounga tonu to maatau whakaaro nui, te punaha QC tino tika; √ 11 tau te mohio ki te kawe i te roopu hoko; √ taiwhanga R&D motuhake; √ E rua nga awheawhe GMP roa kua hainatia; √ He nui nga rawa o nga wheketere mangere mo te kaupapa kua whakaritea; √ He roopu mahi Kairangi me te huarahi rite.Tuhia to korero ki konei ka tukuna mai ki a matou